Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_00551
Ion Channel
Voltage-gated potassium channel subfamily D member 2
Peptide Function
Inhibitor
Gene Name
KCND2
Activity Data (nM)
IC50
13.2 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
YCQKWMWTCDSKRACCEGLRCKLWCRKII
Peptide UniProt Accession
UniParc
UPI0001627736
Peptide Synonyms/Alias
JzTx-V; β/κ-Theraphotoxin-Cg2a; β/κ-TRTX-Cg2a; Peptide F8-15.73; Beta-theraphotoxin-Cj2a
Peptide Species
Chilobrachys guangxiensis (Chinese earth tiger tarantula) (Chilobrachys jingzhao)
Peptide Name
Beta/kappa-theraphotoxin-Cg2a
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−80 mV
Temperature
20–25 °C
Test Method
Patch-clamping
Test Species
Not specified
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available